Publications
2021
STAT3 promotes melanoma metastasis by CEBP-induced repression of the MITF pathway.
Swoboda A,
Soukup R,
Eckel O,
Kinslechner K,
Wingelhofer B,
Schörghofer D,
Sternberg C,
Pham HTT,
Vallianou M,
Horvath J,
Stoiber D,
Kenner L,
Larue L,
Poli V,
Beermann F,
Yokota T,
Kubicek S,
Krausgruber T,
Rendeiro AF,
Bock C,
Zenz R,
Kovacic B,
Aberger F,
Hengstschläger M,
Petzelbauer P,
Mikula M,
Moriggl R.
Oncogene. 2021 Feb;40(6):1091-1105. doi: 10.1038/s41388-020-01584-6. Epub 2020 Dec 15.
2021
Acute BAF perturbation causes immediate changes in chromatin accessibility.
Schick S,
Grosche S,
Kohl KE,
Drpic D,
Jaeger MG,
Marella NC,
Imrichova H,
Lin JG,
Hofstätter G,
Schuster M,
Rendeiro AF,
Koren A,
Petronczki M,
Bock C,
Müller AC,
Winter GE,
Kubicek S.
Nat Genet. 2021 Mar;53(3):269-278. doi: 10.1038/s41588-021-00777-3. Epub 2021 Feb 8.
2021
Precision Medicine in Hematology 2021: Definitions, Tools, Perspectives, and Open Questions.
Valent P,
Orfao A,
Kubicek S,
Staber P,
Haferlach T,
Deininger M,
Kollmann K,
Lion T,
Virgolini I,
Winter G,
Hantschel O,
Kenner L,
Zuber J,
Grebien F,
Moriggl R,
Hoermann G,
Hermine O,
Andreeff M,
Bock C,
Mughal T,
Constantinescu SN,
Kralovics R,
Sexl V,
Skoda R,
Superti-Furga G,
Jäger U.
Hemasphere. 2021 Feb 17;5(3):e536. doi: 10.1097/HS9.0000000000000536. eCollection 2021 Mar.
2021
Publisher Correction: Rational discovery of molecular glue degraders via scalable chemical profiling.
Mayor-Ruiz C,
Bauer S,
Brand M,
Kozicka Z,
Siklos M,
Imrichova H,
Kaltheuner IH,
Hahn E,
Seiler K,
Koren A,
Petzold G,
Fellner M,
Bock C,
Müller AC,
Zuber J,
Geyer M,
Thomä NH,
Kubicek S,
Winter GE.
Nat Chem Biol. 2021 Mar;17(3):361. doi: 10.1038/s41589-021-00735-4.
2021
Hematoxylin binds to mutant calreticulin and disrupts its abnormal interaction with thrombopoietin receptor.
Jia R,
Balligand T,
Atamanyuk V,
Nivarthi H,
Xu E,
Kutzner L,
Weinzierl J,
Nedelec A,
Kubicek S,
Lesyk R,
Zagrijtschuk O,
Constantinescu SN,
Kralovics R.
Blood. 2021 Apr 8;137(14):1920-1931. doi: 10.1182/blood.2020006264.
2020
Age-of-onset information helps identify 76 genetic variants associated with allergic disease.
Ferreira MAR,
Vonk JM,
Baurecht H,
Marenholz I,
Tian C,
Hoffman JD,
Helmer Q,
Tillander A,
Ullemar V,
Lu Y,
Grosche S,
Rüschendorf F,
Granell R,
Brumpton BM,
Fritsche LG,
Bhatta L,
Gabrielsen ME,
Nielsen JB,
Zhou W,
Hveem K,
Langhammer A,
Holmen OL,
Løset M,
Abecasis GR,
Willer CJ,
Emami NC,
Cavazos TB,
Witte JS,
Szwajda A; 23andMe Research Team; collaborators of the SHARE study,
Hinds DA,
Hübner N,
Weidinger S,
Magnusson PK,
Jorgenson E,
Karlsson R,
Paternoster L,
Boomsma DI,
Almqvist C,
Lee YA,
Koppelman GH.
PLoS Genet. 2020 Jun 30;16(6):e1008725. doi: 10.1371/journal.pgen.1008725.
2020
Rational discovery of molecular glue degraders via scalable chemical profiling.
Mayor-Ruiz C,
Bauer S,
Brand M,
Kozicka Z,
Siklos M,
Imrichova H,
Kaltheuner IH,
Hahn E,
Seiler K,
Koren A,
Petzold G,
Fellner M,
Bock C,
Müller AC,
Zuber J,
Geyer M,
Thomä NH,
Kubicek S,
Winter GE.
Nat Chem Biol. 2020 Nov;16(11):1199-1207. doi: 10.1038/s41589-020-0594-x. Epub 2020 Aug 3. Erratum in: Nat Chem Biol. 2021 Mar;17(3):361.
2020
5-Arylidene-2-(4-hydroxyphenyl)aminothiazol-4(5H)-ones with selective inhibitory activity against some leukemia cell lines.
Subtelna I,
Kryshchyshyn-Dylevych A,
Jia R,
Lelyukh M,
Ringler A,
Kubicek S,
Zagrijtschuk O,
Kralovics R,
Lesyk R.
Arch Pharm (Weinheim). 2021 Apr;354(4):e2000342. doi: 10.1002/ardp.202000342. Epub 2020 Nov 25.
2020
STAT3 promotes melanoma metastasis by CEBP-induced repression of the MITF pathway.
Swoboda A,
Soukup R,
Eckel O,
Kinslechner K,
Wingelhofer B,
Schörghofer D,
Sternberg C,
Pham HTT,
Vallianou M,
Horvath J,
Stoiber D,
Kenner L,
Larue L,
Poli V,
Beermann F,
Yokota T,
Kubicek S,
Krausgruber T,
Rendeiro AF,
Bock C,
Zenz R,
Kovacic B,
Aberger F,
Hengstschläger M,
Petzelbauer P,
Mikula M,
Moriggl R.
Oncogene. 2021 Feb;40(6):1091-1105. doi: 10.1038/s41388-020-01584-6.
2020
Pooled protein tagging, cellular imaging, and in situ sequencing for monitoring drug action in real time.
Reicher A,
Koren A,
Kubicek S.
Genome Res. 2020 Dec;30(12):1846-1855. doi: 10.1101/gr.261503.120. Epub 2020 Nov 17.