Publications
2025
Fluorescent PyrAte-(S)-citalopram conjugates enable imaging of the serotonin transporter in living tissue
Oliver J V Belleza,
Iakovos Saridakis,
Nadja K Singer,
Xavier Westergaard,
Sergio Armentia Matheu,
Miran Lemmerer,
Margaux Riomet,
Pedro A Sánchez-Murcia,
Nina Kastner,
Stefanie Rukavina,
Yi Xiao,
Kathrin Jäntsch,
Marco Niello,
Klaus Schicker,
David Sulzer,
Leticia González,
Nuno Maulide,
Harald H Sitte.
Chem Sci. 2025 Mar 3;16(14):6003-6013. doi: 10.1039/d4sc06949h. eCollection 2025 Apr 2.
2024
Probing the Chemical Space of Guanidino-Carboxylic Acids to Identify the First Blockers of the Creatine-Transporter-1
Clemens V Farr,
Yi Xiao,
Ali El-Kasaby,
Manuel Schupp,
Matej Hotka,
Giovanni di Mauro,
Amy Clarke,
Miryam Pastor Fernandez,
Walter Sandtner,
Thomas Stockner,
Christoph Klade,
Nuno Maulide,
Michael Freissmuth.
Mol Pharmacol. 2024 Nov 18;106(6):319-333. doi: 10.1124/molpharm.124.000995.
2024
Diastereoselective hydride transfer enables a synthesis of chiral 1,5-carboxamido-trifluoromethylcarbinols
Roberto Tinelli,
Manuel Schupp,
Immo Klose,
Saad Shaaban,
Boris Maryasin,
Leticia González,
Nuno Maulide.
Chem Sci. 2024 Sep 9;15(38):15751-6. doi: 10.1039/d4sc05049e. Online ahead of print.
2024
Domino Conjugate Addition-1,4-Aryl Migration for the Synthesis of α,β-Difunctionalized Amides
Haoqi Zhang,
Yi Xiao,
Miran Lemmerer,
Tommaso Bortolato,
Nuno Maulide.
JACS Au. 2024 Jun 17;4(7):2456-2461. doi: 10.1021/jacsau.4c00378. eCollection 2024 Jul 22.
2024
PyrAtes: Modular Organic Salts with Large Stokes Shifts for Fluo-rescence Microscopy
Iakovos Saridakis,
Margaux Riomet,
Oliver J V Belleza,
Guilhem Coussanes,
Nadja K Singer,
Nina Kastner,
Yi Xiao,
Elliot Smith,
Veronica Tona,
Aurélien de la Torre,
Eric F Lopes,
Pedro A Sánchez-Murcia,
Leticia González,
Harald H Sitte,
Nuno Maulide.
Angew Chem Int Ed Engl. 2024 May 6;63(19):e202318127. doi: 10.1002/anie.202318127. Epub 2024 Apr 3.
2023
Mechanistic Study on Selenium- and Sulfur-Mediated Isomerization of Hydroxamic Acids
Ricardo Meyrelles,
Manuel Schupp,
Boris Maryasin.
Chemistry. 2023 Dec 19;29(71):e202302386. doi: 10.1002/chem.202302386. Epub 2023 Nov 5.
2022
Synthesis of α-Aryl Acrylamides via Lewis-Base-Mediated Aryl/Hydrogen Exchange
Miran Lemmerer,
Haoqi Zhang,
Anthony J Fernandes,
Tobias Fischer,
Marianne Mießkes,
Yi Xiao,
Nuno Maulide.
Angew Chem Int Ed Engl. 2022 Oct 4;61(40):e202207475. doi: 10.1002/anie.202207475. Epub 2022 Aug 29.
2020
Chemoselective Alpha-Deuteration of Amides via Retro-ene Reaction.
Porte V,
Di Mauro G,
Schupp M,
Kaiser D,
Maulide N.
Chemistry. 2020 Dec 1;26(67):15509-15512. doi: 10.1002/chem.202004103. Epub 2020 Nov 17.
2021
Redox-Neutral Selenium-Catalysed Isomerisation of para-Hydroxamic Acids into para-Aminophenols.
Chuang HY,
Schupp M,
Meyrelles R,
Maryasin B,
Maulide N.
Angew Chem Int Ed Engl. 2021 Mar 24. doi: 10.1002/anie.202100801. Online ahead of print.
2019
A Domino 10-Step Total Synthesis of FR252921 and Its Analogues, Complex Macrocyclic Immunosuppressants.
Chen Y,
Coussanes G,
Souris C,
Aillard P,
Kaldre D,
Runggatscher K,
Kubicek S,
Di Mauro G,
Maryasin B,
Maulide N.
J Am Chem Soc. 2019 Sep 4;141(35):13772-13777. doi: 10.1021/jacs.9b07185.
